2024
Effect of CDC7 inhibition and MYC degradation on neuroendocrine transformation in the lung and prostate cancer.
Quintanal-Villalonga A, Kawasaki K, Redin E, Rakhade S, Durani V, Sabet A, Karthaus W, Zaidi S, Zhan Y, Manoj P, Sridhar H, Zhong H, Mello B, Ciampricotti M, Bhanot U, Haffner M, Socci N, Yu H, Chan J, Rudin C. Effect of CDC7 inhibition and MYC degradation on neuroendocrine transformation in the lung and prostate cancer. Journal Of Clinical Oncology 2024, 42: e20105-e20105. DOI: 10.1200/jco.2024.42.16_suppl.e20105.Peer-Reviewed Original ResearchRisk of transformationNE transformationProstatic adenocarcinomaTherapeutic vulnerabilitiesMYC degradationPhase II clinical trialLung tumor modelDelays tumor relapseII clinical trialsTherapy in vivoIn vivo prostateMechanisms of resistanceMYC isoformsNE phenotypeTumor relapseUntreated tumorsNeuroendocrine transformationProstate cancerStemness transcription factorsPotential therapeutic targetTargeted therapyPoor prognosisTumor modelProstateTumor population
2021
Prostate cancer research in the 21st century; report from the 2021 Coffey‐Holden prostate cancer academy meeting
Miyahira A, Zarif J, Coombs C, Flavell R, Russo J, Zaidi S, Zhao D, Zhao S, Pienta K, Soule H. Prostate cancer research in the 21st century; report from the 2021 Coffey‐Holden prostate cancer academy meeting. The Prostate 2021, 82: 169-181. PMID: 34734426, PMCID: PMC8688282, DOI: 10.1002/pros.24262.Peer-Reviewed Original ResearchConceptsCoffey-Holden Prostate Cancer Academy MeetingCoffey-Holden Prostate Cancer AcademyProstate cancer researchProstate cancerMetastatic castration resistant prostate cancerCastration resistant prostate cancerResistant prostate cancerProstate cancer biologyProstate Cancer FoundationCancer researchAntitumor immunityCancer immunotherapyClonal hematopoiesisMediators of plasticityTumor microenvironmentTargeted therapyProstateCell plasticityCancer FoundationCancer biologyCancerSignaling pathwayCancer genomesSignaling biologyAcademy Meeting
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